5-Bromo-2-methoxypyrimidine synthesis
- Product Name:5-Bromo-2-methoxypyrimidine
- CAS Number:14001-66-2
- Molecular formula:C5H5BrN2O
- Molecular Weight:189.01
124-41-4
698 suppliers
$12.00/25g
32779-36-5
640 suppliers
$5.00/5g
14001-66-2
249 suppliers
$7.00/1g
Yield:14001-66-2 60%
Reaction Conditions:
with methanol at 70;
Steps:
1
Synthesis of Compound 11-3 (0400) To a solution of 11-2 (2.0 g, 10 mmol) in methanol (15 mL) was added CH3ONa (2.16 g, 40 mmol). The resulting mixture was stirred at 70° C. overnight. Methanol was evaporated in vacuum. Water (10 mL) was added carefully to the residue and the mixture was extracted with ethyl acetate (300 mL×3). The combined organic layers were dried over Na2SO4, filtered and concentrated to afford 11-3 as a yellow solid (1.17 g, 60%).
References:
Nivalis Therapeutics, Inc.;Wasley, Jan;Rosenthal, Gary J.;Sun, Xicheng;Strong, Sarah;Qiu, Jian US9138427, 2015, B2 Location in patent:Page/Page column 289-290
67-56-1
751 suppliers
$7.29/5ml-f
38353-06-9
325 suppliers
$15.00/1g
14001-66-2
249 suppliers
$7.00/1g
67-56-1
751 suppliers
$7.29/5ml-f
32779-37-6
190 suppliers
$9.00/1g
14001-66-2
249 suppliers
$7.00/1g
67-56-1
751 suppliers
$7.29/5ml-f
32779-36-5
640 suppliers
$5.00/5g
14001-66-2
249 suppliers
$7.00/1g
14001-67-3
138 suppliers
$8.00/250mg
14001-66-2
249 suppliers
$7.00/1g