ERK Inhibitor

$32 - $228
Product name: ERK Inhibitor
CAS: 1049738-54-6
MF: C14H17ClN2O3S
MW: 328.81
EINECS:
MDL Number:MFCD09038681
Synonyms:(5Z)-3-(2-aminoethyl)-5-[(4-ethoxyphenyl)methylidene]-1,3-thiazolidine-2,4-dione:hydrochloride;ERK Inhibitor - CAS 1049738-54-6 - Calbiochem;3-(2-aminoethyl)-5-[(4-ethoxyphenyl)methylene]-2,4-thiazolidinedione,monohydrochloride;ERK-IN-4

Price4 Properties Safety Information Description

4 prices

Selected condition：

Brand

AK Scientific
Cayman Chemical

Package

500μg
1mg
5mg

ManufacturerAK Scientific
Product number9473CW
Product descriptionErkInhibitor
Packaging5mg
Price$228
Updated2021-12-16
Buy

ManufacturerCayman Chemical
Product number15944
Product descriptionERK Inhibitor ≥95%
Packaging500μg
Price$32
Updated2024-03-01
Buy

ManufacturerCayman Chemical
Product number15944
Product descriptionERK Inhibitor ≥95%
Packaging1mg
Price$50
Updated2024-03-01
Buy

ManufacturerCayman Chemical
Product number15944
Product descriptionERK Inhibitor ≥95%
Packaging5mg
Price$117
Updated2024-03-01
Buy

Manufacturer	Product number	Product description	Packaging	Price	Updated	Buy
AK Scientific	9473CW	ErkInhibitor	5mg	$228	2021-12-16	Buy
Cayman Chemical	15944	ERK Inhibitor ≥95%	500μg	$32	2024-03-01	Buy
Cayman Chemical	15944	ERK Inhibitor ≥95%	1mg	$50	2024-03-01	Buy
Cayman Chemical	15944	ERK Inhibitor ≥95%	5mg	$117	2024-03-01	Buy

Properties

storage temp. :+2C to +8C
solubility :DMSO: 2 mg/ml
form :Light yellow solid
color :Off-white to yellow

Safety Information

Symbol(GHS):

Signal word:

Hazard statements:

Code	Hazard statements	Hazard class	Category	Signal word	Pictogram	P-Codes

Precautionary statements:

Description

ERK inhibitor is a cell-permeable inhibitor that binds ERK2 near its docking domain (KD = 5 μM). This prevents its interaction with protein substrates without inhibiting catalytic activity. ERK inhibitor blocks ERK-specific phosphorylation of ribosomal S6 kinase-1 and ternary complex factor Elk-1 but does not affect ERK1/2 phosphorylation by MEK1/2. Presumably through its effects on ERK, ERK inhibitor completely prevents proliferation of HeLa cells (IC50 = 15-20 μM), A549 lung carcinoma cells (IC50 = 25 μM), Sum-159 estrogen receptor-negative breast cancer cells and HT1080 fibrosarcoma cells.

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