Cetilistat
- $5 - $750
- Product name: Cetilistat
- CAS: 282526-98-1
- MF: C25H39NO3
- MW: 401.58
- EINECS:1308068-626-2
- MDL Number:MFCD09839697
- Synonyms:cetilistat;Cetilistat(Alt-962);Cetilstat;2-(Hexadecycloxy)-6-methyl-4H-3,1-benzoxazin-4-one;4H-3,1-Benzoxazin-4-one,2-(hexadecyloxy)-6-Methyl-;Xinli orlistat;2-hexadecoxy-6-methyl-3,1-benzoxazin-4-one;Cetilistat (ATL-962)
29 prices
Selected condition:
Brand
- AK Scientific
- Ambeed
- American Custom Chemicals Corporation
- ApexBio Technology
- Arctom
- Biosynth Carbosynth
- Chem-Impex
- Crysdot
- CSNpharm
- Labseeker
- TCI Chemical
- TRC
- Usbiological
Package
- 50mg
- 100mg
- 200mg
- 250mg
- 500mg
- 1g
- 5g
- 10g
- 25g
- 50g
- 100g
- 250g
- 1kg
- ManufacturerAK Scientific
- Product numberJ51544
- Product descriptionCitilistat
- Packaging5g
- Price$25
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA117014
- Product descriptionCetilistat 98+%
- Packaging1g
- Price$13
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA117014
- Product descriptionCetilistat 98+%
- Packaging5g
- Price$23
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA117014
- Product descriptionCetilistat 98+%
- Packaging10g
- Price$37
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA117014
- Product descriptionCetilistat 98+%
- Packaging25g
- Price$69
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0002040
- Product descriptionCITILISTAT 95.00%
- Packaging1G
- Price$178.5
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberC7022
- Product descriptionCetilistat
- Packaging200mg
- Price$45
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberC7022
- Product descriptionCetilistat
- Packaging500mg
- Price$65
- Updated2021-12-16
- Buy
- ManufacturerArctom
- Product numberAS437583
- Product descriptionCetilistat ≥98%
- Packaging250mg
- Price$5
- Updated2021-12-16
- Buy
- ManufacturerArctom
- Product numberAS437583
- Product descriptionCetilistat ≥98%
- Packaging1g
- Price$13
- Updated2021-12-16
- Buy
- ManufacturerArctom
- Product numberAS437583
- Product descriptionCetilistat ≥98%
- Packaging5g
- Price$23
- Updated2021-12-16
- Buy
- ManufacturerArctom
- Product numberAS437583
- Product descriptionCetilistat ≥98%
- Packaging10g
- Price$37
- Updated2021-12-16
- Buy
- ManufacturerArctom
- Product numberAS437583
- Product descriptionCetilistat ≥98%
- Packaging25g
- Price$68
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberFH16224
- Product descriptionCetilistat
- Packaging10g
- Price$45
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberBC166233
- Product descriptionCetilistat
- Packaging100mg
- Price$50
- Updated2021-12-16
- Buy
- ManufacturerBiosynth Carbosynth
- Product numberFH16224
- Product descriptionCetilistat
- Packaging25g
- Price$70
- Updated2021-12-16
- Buy
Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
---|---|---|---|---|---|---|
AK Scientific | J51544 | Citilistat | 5g | $25 | 2021-12-16 | Buy |
Ambeed | A117014 | Cetilistat 98+% | 1g | $13 | 2021-12-16 | Buy |
Ambeed | A117014 | Cetilistat 98+% | 5g | $23 | 2021-12-16 | Buy |
Ambeed | A117014 | Cetilistat 98+% | 10g | $37 | 2021-12-16 | Buy |
Ambeed | A117014 | Cetilistat 98+% | 25g | $69 | 2021-12-16 | Buy |
American Custom Chemicals Corporation | API0002040 | CITILISTAT 95.00% | 1G | $178.5 | 2021-12-16 | Buy |
ApexBio Technology | C7022 | Cetilistat | 200mg | $45 | 2021-12-16 | Buy |
ApexBio Technology | C7022 | Cetilistat | 500mg | $65 | 2021-12-16 | Buy |
Arctom | AS437583 | Cetilistat ≥98% | 250mg | $5 | 2021-12-16 | Buy |
Arctom | AS437583 | Cetilistat ≥98% | 1g | $13 | 2021-12-16 | Buy |
Arctom | AS437583 | Cetilistat ≥98% | 5g | $23 | 2021-12-16 | Buy |
Arctom | AS437583 | Cetilistat ≥98% | 10g | $37 | 2021-12-16 | Buy |
Arctom | AS437583 | Cetilistat ≥98% | 25g | $68 | 2021-12-16 | Buy |
Biosynth Carbosynth | FH16224 | Cetilistat | 10g | $45 | 2021-12-16 | Buy |
Biosynth Carbosynth | BC166233 | Cetilistat | 100mg | $50 | 2021-12-16 | Buy |
Biosynth Carbosynth | FH16224 | Cetilistat | 25g | $70 | 2021-12-16 | Buy |
Properties
Melting point :72.0 to 76.0 °C
Boiling point :509.7±43.0 °C(Predicted)
Density :1.02
storage temp. :2-8°C
solubility :Chloroform (Slightly), Ethyl Acetate (Slightly)
form :Solid
pka :2.96±0.20(Predicted)
color :White to Off-White
InChI :InChI=1S/C25H39NO3/c1-3-4-5-6-7-8-9-10-11-12-13-14-15-16-19-28-25-26-23-18-17-21(2)20-22(23)24(27)29-25/h17-18,20H,3-16,19H2,1-2H3
InChIKey :MVCQKIKWYUURMU-UHFFFAOYSA-N
SMILES :N1C2=CC=C(C)C=C2C(=O)OC=1OCCCCCCCCCCCCCCCC
CAS DataBase Reference :282526-98-1(CAS DataBase Reference)
Boiling point :509.7±43.0 °C(Predicted)
Density :1.02
storage temp. :2-8°C
solubility :Chloroform (Slightly), Ethyl Acetate (Slightly)
form :Solid
pka :2.96±0.20(Predicted)
color :White to Off-White
InChI :InChI=1S/C25H39NO3/c1-3-4-5-6-7-8-9-10-11-12-13-14-15-16-19-28-25-26-23-18-17-21(2)20-22(23)24(27)29-25/h17-18,20H,3-16,19H2,1-2H3
InChIKey :MVCQKIKWYUURMU-UHFFFAOYSA-N
SMILES :N1C2=CC=C(C)C=C2C(=O)OC=1OCCCCCCCCCCCCCCCC
CAS DataBase Reference :282526-98-1(CAS DataBase Reference)
Safety Information
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Description
Cetilistat (also known as ATL-962) was approved in September 2013 by the Japanese Ministry of Health, Labor and Welfare for the treatment of obesity, limited to patients with both type 2 diabetes mellitus (T2DM) and dyslipidemia, and with a body mass index (BMI)25 kg/m2 in spite of dietary treatment and/or exercise therapy. As with orlistat, cetilistat works via inhibition of pancreatic lipases in the gut to inhibit fat absorption and thereby reduce caloric uptake from diet. The medicinal chemistry program has not been described in the scientific literature, but the patent describing cetilistat also describes the synthesis of analogs with varied aryl substituents and lipophilic tails. The synthesis of cetilistat involves condensation of a hexadecylcarbonochloridate with 2-amino-5-methylbenzoic acid; other analogs were synthesized by varying the carbonochloridate and 2-aminobenzoic acid components. Cetilistat is a potent inhibitor of human and rat pancreatic lipase with IC50s of 15 and 136 nM, respectively, with little inhibition of trypsin or chymotrypsin.Related product price
- Paraquat dichloride
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$9-7620
Suppliers and manufacturers
Wuhan Mayue Longteng Technology Development Co., Ltd.
Apeloa production Co.,Limited
Shandong Hanjiang Chemical Co., Ltd
Shanghai Likang New Materials Co., Limited