8-HYDROXY-2H-BENZO[B][1,4]OXAZIN-3(4H)-ONE synthesis
- Product Name:8-HYDROXY-2H-BENZO[B][1,4]OXAZIN-3(4H)-ONE
- CAS Number:258532-76-2
- Molecular formula:C8H7NO3
- Molecular Weight:165.15
107-83-5
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Yield: 70%
Reaction Conditions:
in ethyl acetate
Steps:
70.1 8-(2-{[3-(1-Piperazinyl)-2-pyrazinyl]oxy}ethoxy)-2H-1,4-benzoxazin-3(4H)-one, Maleate
Step 1: 8-Hydroxy-2H-1,4-benzoxazin-3(4H)-one. The title compound was prepared according to procedure described in J Med. Chem. 1996, 39, 3533-3538 by replacing 2-amino-m-cresol with 3-amino-pyrocatechol. *The crude product was purified by column chromatography on silica gel using EtOAc/isohexane (1:2 to 2:1) as eluent. Solid; yield 70%. MS m/z 165 (M)+. Anal. (C8H7NO3) C, H, N.
References:
Biovitrum AB US6465467, 2002, B1
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