2-Bromo-3-hydroxypyridine synthesis
- Product Name:2-Bromo-3-hydroxypyridine
- CAS Number:6602-32-0
- Molecular formula:C5H4BrNO
- Molecular Weight:174
24100-18-3
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$6.00/1g
6602-32-0
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$10.00/1g
Yield:6602-32-0 94%
Reaction Conditions:
with hydrogen bromide in dichloromethane at 140;Inert atmosphere;
Steps:
2-Bromo-3-hydroxypyridine (22b)
2-bromo-3-methoxypyridine (295 mg, 1.57 mmol) was heated in hydrobromide acid (5 ml) to 140 °C and stirred overnight. The solution was neutralized with a saturated sodium bicarbonate solution and extracted three times with ethyl acetate. The combined organic layers were dried over Na2SO4 and the solvent was removed under reduced pressure. Yield: 258 mg (94 %), white crystals. 1H-NMR((CD3)2CO, 500 MHz): δH = 9.26 (s, 1H), 7.89 (dd, J = 1.6, 4.4 Hz, 1H), 7.32-7.36 (m,1H), 7.23-7.27 (m, 1H); 13C-NMR ((CD3)2CO, 125 MHz): δC = 152.4, 142.1, 131.9, 125.3, 124.5.
References:
Hu, Qingzhong;Kunde, Jessica;Hanke, Nina;Hartmann, Rolf W. [European Journal of Medicinal Chemistry,2015,vol. 96,p. 139 - 150] Location in patent:supporting information
109-00-2
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$10.00/10g
6602-32-0
413 suppliers
$10.00/1g
109-00-2
590 suppliers
$10.00/10g
6602-32-0
413 suppliers
$10.00/1g
6602-33-1
107 suppliers
$14.00/250mg
109-00-2
590 suppliers
$10.00/10g
6602-32-0
413 suppliers
$10.00/1g
6602-33-1
107 suppliers
$14.00/250mg
6602-34-2
51 suppliers
$120.00/1g
109-00-2
590 suppliers
$10.00/10g
6602-32-0
413 suppliers
$10.00/1g
6602-33-1
107 suppliers
$14.00/250mg
129611-31-0
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