1-(3-Cyanopyridyl-2)-2-Phenyl-4-Methylpyperazine synthesis
- Product Name:1-(3-Cyanopyridyl-2)-2-Phenyl-4-Methylpyperazine
- CAS Number:61337-88-0
- Molecular formula:C17H18N4
- Molecular Weight:278.35
6602-54-6
494 suppliers
$6.00/10g
5271-27-2
249 suppliers
$15.00/1g
61338-13-4
135 suppliers
$41.00/100mg
61337-88-0
45 suppliers
inquiry
Yield:-
Reaction Conditions:
potassium fluoride;N,N-dimethyl-formamide
Steps:
5 Preparation of 1,2,3,4,10,14b-hexahydro-2-methyl-pyrazino[2,1-a] pyrido{2,3-c} [2]Benzazepine of Formula 17:
EXAMPLE-5 Preparation of 1,2,3,4,10,14b-hexahydro-2-methyl-pyrazino[2,1-a] pyrido{2,3-c} [2]Benzazepine of Formula 17: 1-Methyl-3-phenylpiperazine (50.0 g, 0.284 mol) was heated with 2-chloro-3-cyanopyridine (39.35 g, 0.284 mol) in the presence of potassium fluoride (49.51 g, 0.852 mol) and N,N-dimethylformamide (750.0 ml) as a solvent for 30.0 hrs at 148-154° C., followed by quenching with water and extraction with ethyl acetate gave 1-(3-cyanopyridyl-2-)-4-methyl-2-phenylpiperazine (70.0 g). 1-(3-Cyanopyridyl-2)-4-methyl-2-phenylpiperazine on hydrolysis with saturated alcoholic potassium hydroxide solution (850.0 ml) at 80-85° C. followed by extraction with chloroform gave 1-(3-carboxypyridyl-2)-4-methyl-2-phenylpiperazine (20.0 g).
References:
Sebastian, Sonny;Patel, Hetal Virendra;Thennati, Rajamannar US2002/95038, 2002, A1
6602-54-6
494 suppliers
$6.00/10g
821-55-6
330 suppliers
$7.00/25g
5271-27-2
249 suppliers
$15.00/1g
61337-88-0
45 suppliers
inquiry
6602-54-6
494 suppliers
$6.00/10g
5271-27-2
249 suppliers
$15.00/1g
1000210-73-0
0 suppliers
inquiry
61337-88-0
45 suppliers
inquiry