中文名:AT7519,CDK抑制劑
英文名:AT7519
英文別名:AT7519|844442-38-2|AT-7519|4-(2,6-dichlorobenzamido)-N-(piperidin-4-yl)-1H-pyrazole-3-carboxamide|AT 7519|AT7519 Hydrochloride|4-(2,6-Dichloro-benzoylamino)-1H-pyrazole-3-carboxylic acid piperidin-4-ylamide|Cdki at7519|N-(4-Piperidinyl)-4-(2,6-dichloroben
純度:≥99%
貨號(hào):A127001
包裝:100mg、25mg、5mg
Cas號(hào):844442-38-2
存儲(chǔ)溫度:-20°C儲(chǔ)存
產(chǎn)品介紹:
AT7519是多種CDK抑制劑,作用于CDK1, 2, 4, 6和9時(shí),IC50為10-210 nM,對(duì)CDK3作用效果稍弱,對(duì)CDK7幾乎沒有抑制活性。Phase 2。A novel small molecule effective as a pan-Cdk inhibitor for Cdk1, Cdk2, Cdk3, Cdk4, Cdk5 and Cdk6.
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