Enzastaurin (LY317615)
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Enzastaurin (LY317615) ??
- ???
- 249-261℃
- ?? ?
- 767.2±60.0 °C(Predicted)
- ??
- 1.34
- RTECS ??
- UX9626850
- ???
- 417.8℃
- ?? ??
- -20°C
- ???
- DMSO: ???10mg/mL, ??(??)
- ??? ??
- ??
- ?? ?? (pKa)
- 7.88±0.60(Predicted)
- ??
- , ?? ????? ?? ???-?????
- ???
- ??? ?? ?????? 1? ?? ??????. DMSO ??? -20°C?? ?? 3?? ?? ??? ? ????.
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- ?? ? ???? ?? (GHS)
Enzastaurin (LY317615) C??? ??, ??, ??
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PKCβ-selective inhibitor, suppresses angiogenesis.Biochem/physiol Actions
Enzastaurin is a potent and PKCβ preferring inhibitor. Also, Enzastaurin inhibits AKT and GSK3β. Enzastaurin acts as anti-angiogenic and antineoplastic agent.Enzastaurin (LY317615) ?? ?? ? ???
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Enzastaurin (LY317615) ?? ??
???( 169)?? ??
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Capot Chemical Co.,Ltd. | +86-(0)57185586718 +86-13336195806 |
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