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PF-4800567 HCl

PF-4800567 HCl ??? ???
?? ??:
1391052-28-0
???:
PF-4800567 HCl
???(??):
PF-4800567 HCl;PF-4800567 hydrochloride >=98% (HPLC);3-[(3-chlorophenoxy)methyl]-1-(oxan-4-yl)pyrazolo[3,4-d]pyrimidin-4-amine:hydrochloride
CBNumber:
CB13145563
???:
C17H19Cl2N5O2
??? ??:
396.27
MOL ??:
1391052-28-0.mol
MSDS ??:
SDS

PF-4800567 HCl ??

?? ??
Desiccate at RT
???
Soluble to 100 mM in DMSO
??? ??
??
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white to beige

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PF-4800567 HCl C??? ??, ??, ??

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PF 4800567 is a selective casein kinase 1ε inhibitor; displays 22-fold greater potency towards CK1ε than CK1δ (IC50 values are 32 and 711 nM for CK1ε and CK1δ respectively). ATP competitive. Displays minimal effect on the circadian clock.

PF-4800567 HCl ?? ?? ? ???

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PF-4800567 HCl ?? ??

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