NALOXONE BENZOYLHYDRAZONE Chemische Eigenschaften,Einsatz,Produktion Methoden
Biologische Aktivit?t
Mixed opioid receptor agonist/antagonist. Acts as a potent and full agonist at κ , and a partial agonist at μ and δ opioid receptors (pEC 50 values are 9.45, 8.74 and 8.61 in a cAMP assay, 9.70, 8.59 and 8.49 in a [ 35 S]GTP γ S binding assay respectively). Fails to exert agonist effects at NOP receptors and antagonizes agonist-induced NOP activation. Stimulates κ -, μ - and δ -mediated analgesia and blocks NOP-induced supraspinal nociception.
NALOXONE BENZOYLHYDRAZONE Upstream-Materialien And Downstream Produkte
Upstream-Materialien
Downstream Produkte