methylnaltrexone Chemische Eigenschaften,Einsatz,Produktion Methoden

Allgemeine Beschreibung

Methylnaltrexone (Relistor) is the methylated, quaternaryform of naltrexone . The permanently chargednitrogen prevents the drug from crossing the blood-brainbarrier. Thus, it only acts as an antagonist at peripheralopioid receptors. Relistor was approved in April 2008 totreat opioid-induced constipation in patients receiving palliativecare. It is administered as a SC injection once everyother day.

methylnaltrexone Upstream-Materialien And Downstream Produkte

Upstream-Materialien

Downstream Produkte

methylnaltrexone Anbieter Lieferant Produzent Hersteller Vertrieb H?ndler.

Firmenname	Telefon	E-Mail	Land	Produktkatalog	Edge Rate
TargetMol Chemicals Inc.	+8613564774135	zijue.cai@tsbiochem.com	United States	19885	58
QUALITY CONTROL SOLUTIONS LTD.	0755-66853366; 13670046396	ORDERS@QCSRM.COM	China	24342	58
TargetMol Chemicals Inc.	15002134094	marketing@targetmol.cn	China	19704	58

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• methylnaltrexone
• 17-(Cyclopropylmethyl)-4,5α-epoxy-3-methoxy-14-hydroxymorphinan-6-one
• 3-Methoxy-14-hydroxy-17-(cyclopropylmethyl)-4,5α-epoxymorphinan-6-one
• 3-O-Methylnaltrexone
• 4,5α-Epoxy-3-methoxy-14β-hydroxy-17-(cyclopropylmethyl)morphinan-6-one
• Naltrexone methyl ether
• 17-(Cyclopropylmethyl)-4,5alpha-epoxy-3,14-dihydroxy-17-methyl-6-oxomorphinanium
• 17-(Cyclopropylmethyl)-4,5-epoxy-3,14-dihydroxymorphinanium-6-one
• Methylnaltrexonium
• Morphinanium, 17-(cyclopropylmethyl)-4,5-epoxy-3,14-dihydroxy-17-methyl-6-oxo-, (5alpha)-
• Mrz 2663
• Mrz-2663
• Naltrexone mb
• N-Methylnaltrexone
• 83387-25-1