Identification | Back Directory | [Name]
R-IMPP | [CAS]
2133832-83-2 | [Synonyms]
R-IMPP Benzenepropanamide, N-1-isoquinolinyl-4-methoxy-N-(3R)-3-piperidinyl- | [Molecular Formula]
C24H27N3O2 | [MDL Number]
MFCD31544323 | [MOL File]
2133832-83-2.mol | [Molecular Weight]
389.49 |
Chemical Properties | Back Directory | [Boiling point ]
594.4±50.0 °C(Predicted) | [density ]
1.186±0.06 g/cm3(Predicted) | [storage temp. ]
Store at -20°C | [solubility ]
DMF: 1 mg/ml; DMSO: 10 mg/ml | [form ]
A crystalline solid | [pka]
9.14±0.10(Predicted) | [color ]
Light yellow to yellow |
Hazard Information | Back Directory | [Description]
(R)-IMPP is a cell-permeable inhibitor of the secretion of proprotein convertase subtilisin/kexin type 9 (PCSK9; IC50 = 4.8 μM). It promotes the uptake of LDL cholesterol in hepatoma cells by increasing LDL receptor levels. (R)-IMPP apparently impairs PCSK9 secretion by causing transcript-dependent inhibition of PCSK9 translation. | [storage]
Store at -20°C |
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DC Chemicals
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