3-Iodo-1H-pyrazolo[3,4-d]pyrimidin-4-amine synthesis
- Product Name:3-Iodo-1H-pyrazolo[3,4-d]pyrimidin-4-amine
- CAS Number:151266-23-8
- Molecular formula:C5H4IN5
- Molecular Weight:261.02
516-12-1
539 suppliers
$5.00/5g
2380-63-4
366 suppliers
$9.00/1g
151266-23-8
330 suppliers
$22.00/1g
Yield:151266-23-8 86%
Reaction Conditions:
in N,N-dimethyl-formamide at 80; for 12 h;
Steps:
1.1 synthesis of 3-iodo-1H-Pyrazolo[3, 4-d] pyrimidine-4-amine
Pyrazolo [3,4-d] pyrimidin-4-amine (15.0 g, 111.1 mmol) was dissolved in DMF (150 mL) N-iodosuccinimide (37.5 g, 166. 6 mmol) was slowly added to the reaction mixture, and the reaction was stirred at 80 ° C for 12 h. stopWater (40 mL) was added to the reaction mixture, and the mixture was suction filtered. The solid was washed with water (80 mL), ethanol (60 mL) and dried to give to a yellow solid (24. 9 g, 86%).
References:
Guangdong HEC Pharmaceutical Co., Ltd;LIU, BING;BAI, SHUN;ZHANG, YINGJUN;ZHENG, CHANGCHUN;YANG, TIPING;ZHOU, YOUBAI CN105399756, 2016, A Location in patent:Paragraph 0155; 0165-0166
2380-63-4
366 suppliers
$9.00/1g
151266-23-8
330 suppliers
$22.00/1g
64834-00-0
8 suppliers
inquiry
151266-23-8
330 suppliers
$22.00/1g
5399-92-8
232 suppliers
$13.43/250mgs:
151266-23-8
330 suppliers
$22.00/1g