價格 | ¥15300 | ¥11700 | ¥19500 |
包裝 | 50mg | 25mg | 100mg |
最小起訂量 | 1mg |
發(fā)貨地 | 上海 |
更新日期 | 2025-02-28 |
中文名稱:化合物 DHMEQ racemate | 英文名稱:DHMEQ racemate |
CAS:287194-38-1 | 品牌: TargetMol |
產地: 美國 | 保存條件: Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
產品類別: 抑制劑 | |
貨號: T11018 |
名稱 | DHMEQ racemate |
描述 | DHMEQ racemate is an NF-κB inhibitor. The activity of DHMEQ racemate is lower than (-)-DHMEQ. |
體外活性 | DHMEQ racemate (DHM3EQ) and (-)-DHMEQ (DHM2EQ) inhibit TNF-a-induced NF-kB activation. (-)-DHMEQ is more effective and less toxic than DHMEQ racemate. |
體內活性 | The anti-arthritis effect of (-)-DHMEQ (DHM2EQ) and DHMEQ racemate (DHM3EQ) on type II collagen-induced arthritis in DBA1/J mice was studied. Because of its pathological similarity to human rheumatoid arthritis, this animal model is widely used to evaluate anti-rheumatic drugs. Cause arthritis and score it. (-)-DHMEQ significantly inhibited type II collagen-induced arthritis in mice, while DHMEQ racemates tended to only slightly inhibit it. |
存儲條件 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
溶解度 | DMSO : 32 mg/mL (122.50 mM) |
關鍵字 | DHMEQ racemate |
相關產品 | Lidocaine hydrochloride | sodium lauroyl-α-hydroxyethyl sulfonate | Sodium Houttuyfonate | Lidocaine | Caffeic Acid Phenethyl Ester | 5-Aminosalicylic Acid | Diallyl disulfide | Glucosamine | Sodium salicylate | Zingerone | Indole-3-carbinol | Diethylmaleate |
成立日期 | 2013-04-18 (12年) | 注冊資本 | 566.265100萬人民幣 |
員工人數 | 100-500人 | 年營業(yè)額 | ¥ 1億以上 |
主營行業(yè) | 天然產物,生化試劑,分子生物學,分子砌塊,生物技術服務 | 經營模式 | 貿易,工廠,試劑,定制,服務 |
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