Molecular Formula:
C59H84N16O12
Relative Molecular Mass:
1209.5 (net)
CAS-Number:
53714-56-0 (net), 74381-53-6 (acetate)
Synonyms:
Leuprorelin; (Des-Gly10,D-Leu6,Pro-NHEt9)-LHRH
Sequence:
Pyr-His-Trp-Ser-Tyr-D-Leu-Leu-Arg-Pro-NHEt acetate salt
Fields of Application:
Advanced hormone-dependent prostate cancer
Advanced hormone-dependent breast cancer
Endometriosis
Uterine myoma
Central precocious puberty
Active Substance:
Leuprolide Acetate is a potent LHRH (GnRH) agonist. After a transient increase, continuous
administration of leuprolide,results in downregulation of LH and FSH levels followed bya suppression of ovarian and testicular steroid biosynthesis.
Studies with female Alzheimer patients indicate that application of leuprolide acetate in
combination with an acetylcholinesterase inhibitor stabilizes the cognitive functions in mild-to-moderate cases.
關(guān)鍵字: 亮丙瑞林;醋酸亮丙瑞林;Leuprolide Acetate;Leuprolide