生物活性Amastatinhydrochloride是一種緩慢,緊密結(jié)合的競爭性氨肽酶(AP)抑制劑,對氣單胞菌氨肽酶,胞質(zhì)亮氨酸氨肽酶,微粒體氨肽酶的Ki值分別為0.26nM,30nM,52nM。體外研究Amastatinhydrochloride(1-10000ng/ml)exhibitcdinhibitoryprofilesofE.cuniczclireplicationinvitroinadosedependentmanner.
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