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TG003

  Cat. No.:  DC8932   Featured
Chemical Structure
300801-52-9
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More than 5000 active chemicals with high quality for research!
Field of application
TG003 is a potent and ATP-competitive Cdc2-like kinase (Clk) inhibitor with IC50 of 20 nM, 200 nM, and 15 nM for Clk1, Clk2, and Clk4, respectively. No inhibitory effect on Clk3, SRPK1, SRPK2, or PKC.
Cas No.: 300801-52-9
Chemical Name: (Z)-1-(3-Ethyl-5-methoxy-2,3-dihydrobenzothiazol-2-ylidene)propan-2-one
Synonyms: 2-Propanone,1-(3-ethyl-5-methoxy-2(3H)-benzothiazolylidene)-;(Z)-1-(3-Ethyl-5-methoxybenzo[d]thiazol-2(3H)-ylidene)propan-2-one;1-(3-ethyl-5-methoxy-2(3H)-benzothiazolylidene)-2-Propanone;CDC2-LIKE KINASE INHIBITOR, TG003;TG003;(1Z)-1-(3-Ethyl-5-methoxy-1,3-benzothiazol-2(3H)-ylidene)acetone;(1Z)-1-(3-Ethyl-5-methoxy-1,3-benzothiazol-2-ylidene)propan-2-one;2-Propanone, 1-(3-ethyl-5-methoxy-2(3H)-benzothiazolylidene)-, (1Z)-;(Z)-1-(3-Ethyl-5-methoxy-2,3-dihydrobenzothiazol-2-ylidene)propan-2-one;TG 003;Cdc2-Like kinase inhibitor;Clk inhibitor;Clk Inhibitor, TG003;MLS000077198;GTPL5942
SMILES: COC1C=C2N(CC)\C(=C\C(C)=O)SC2=CC=1
Formula: C13H15NO2S
M.Wt: 249.3287
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: TG003 is a potent and ATP-competitive Cdc2-like kinase (Clk) inhibitor with IC50 of 20 nM, 200 nM, and 15 nM for Clk1, Clk2, and Clk4, respectively. No inhibitory effect on Clk3, SRPK1, SRPK2, or PKC.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
2018-0101
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