成人免费xx,国产又黄又湿又刺激不卡网站,成人性视频app菠萝网站,色天天天天

  2. GPCR/G Protein Neuronal Signaling Metabolic Enzyme/Protease
  3. Adrenergic Receptor Renin 5-HT Receptor
  4. Bopindolol (malonate)

Bopindolol (malonate)  (Synonyms: 波吲洛爾丙二酸鹽; (±)-Bopindolol (malonate))

目錄號(hào): HY-B1562B
產(chǎn)品使用指南 技術(shù)支持

Bopindolol ((±)-Bopindolol) malonate 是一種口服活性的 β-腎上腺素受體 (ARs) 拮抗劑，具有部分激動(dòng)劑活性。Bopindolol malonate 對(duì) β1-和 β2-ARs 無(wú)選擇性，對(duì) β3-AR 亞型親和力低。Bopindolol malonate 具有內(nèi)在擬交感神經(jīng)和膜穩(wěn)定作用，抑制腎素 (renin) 分泌，并與 5-HT 受體相互作用。Bopindolol malonate 是 Pindolol (HY-B0982) 的前體活性分子，可用于原發(fā)性和腎血管性高血壓的研究。

MCE 的所有產(chǎn)品僅用作科學(xué)研究或藥證申報(bào)，我們不為任何個(gè)人用途提供產(chǎn)品和服務(wù)

Bopindolol (malonate) Chemical Structure

Bopindolol (malonate) Chemical Structure

CAS No. : 82857-38-3

1.  客戶無(wú)需承擔(dān)相應(yīng)的運(yùn)輸費(fèi)用。

2.  同一機(jī)構(gòu)（單位）同一產(chǎn)品試用裝僅限申領(lǐng)一次，同一機(jī)構(gòu)（單位）一年內(nèi)

     可免費(fèi)申領(lǐng)三個(gè)不同產(chǎn)品的試用裝。

3.  試用裝只面向終端客戶。

規(guī)格 價(jià)格 是否有貨 數(shù)量
25 mg ￥754
3 - 4 周
50 mg ￥1203
3 - 4 周
100 mg ￥1922
3 - 4 周
200 mg   詢價(jià)  
500 mg   詢價(jià)  

* Please select Quantity before adding items.

Customer Review

Other Forms of Bopindolol (malonate):

  • 生物活性

  • 純度 & 產(chǎn)品資料

  • 參考文獻(xiàn)

生物活性

Bopindolol ((±)-Bopindolol) malonate is an orally active antagonist of β-adrenoceptors (ARs) with partial agonist activity. Bopindolol malonate is non-selective for β1- and β2-ARs and has low affinity for β3-AR subtype. Bopindolol malonate has intrinsic sympathomimetic as well as membrane stabilizing actions, inhibits renin secretion, and interacts with 5-HT receptors. Bopindolol malonate is a proagent of Pindolol (HY-B0982). Bopindolol malonate can be used for essential and renovascular hypertension research.

IC50 & Target

Adrenergic receptor, Renin, 5-HT receptors[1][4]
體內(nèi)研究
(In Vivo)

Bopindolol (intravenous injection; 8, 16 and 32 μg/kg) causes a dose-dependent inhibition of isoprenaline-induced tachycardia, and this agent is 4 times more potent than propranolol in anaesthetised dogs[1].
Bopindolol (0.3, 1 and 3 mg/kg; IP; single dosage) produces dose dependent decreases in diastolic blood pressure and in heart rate[2].

MCE has not independently confirmed the accuracy of these methods. They are for reference only.

Animal Model: Male Wistar rats (260-300 g)[2]
Dosage: 0.3, 1 and 3 mg/kg
Administration: IP; single dosage
Result: Produced dose dependent decreases in diastolic blood pressure, and the decrease of about 8 mmHg at 3 mg/kg.
Decreased the heart rate in a dose-dependent manner.
分子量

484.54

Formula

C26H32N2O7
CAS 號(hào)
中文名稱

波吲洛爾丙二酸鹽；吲苯脂心安丙二酸鹽
運(yùn)輸條件

Room temperature in continental US; may vary elsewhere.
儲(chǔ)存方式

Please store the product under the recommended conditions in the Certificate of Analysis.
純度 & 產(chǎn)品資料
參考文獻(xiàn)

  • 摩爾計(jì)算器

  • 稀釋計(jì)算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

質(zhì)量   濃度   體積   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

濃度 (start) × 體積 (start) = 濃度 (final) × 體積 (final)
× = ×
C1   V1   C2   V2
Help & FAQs
  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

您最近查看的產(chǎn)品:

Your information is safe with us. * Required Fields.

   產(chǎn)品名稱：

  

* 需求量：

* 客戶姓名：

 

* Email：

* 電話：

 

* 公司或機(jī)構(gòu)名稱：

   留言給我們：

Bulk Inquiry

Inquiry Information

產(chǎn)品名稱：
Bopindolol (malonate)
目錄號(hào)：
HY-B1562B
需求量：