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  1. Metabolic Enzyme/Protease
  2. Drug Metabolite
  3. Cinacalcet metabolite M4

Cinacalcet metabolite M4 是 Cinacalcet 的代謝物。Cinacalcet 是一種可口服的 Ca receptor (CaR) 激動(dòng)劑,用于心血管疾病。

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Cinacalcet metabolite M4 Chemical Structure

Cinacalcet metabolite M4 Chemical Structure

CAS No. : 104774-87-0

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  • 生物活性

  • 純度 & 產(chǎn)品資料

  • 參考文獻(xiàn)

生物活性

Cinacalcet metabolite M4 is a metabolite of Cinacalcet. Cinacalcet is an orally active, allosteric agonist of Ca receptor (CaR), used for cardiovascular disease[1][2].

分子量

203.20

Formula

C10H12F3N

CAS 號(hào)
性狀

液體(密度:1.154±0.06 g/cm3

顏色

Colorless to light yellow

運(yùn)輸條件

Room temperature in continental US; may vary elsewhere.

儲(chǔ)存方式
Pure form -20°C 3 years
4°C 2 years
In solvent -80°C 6 months
-20°C 1 month
純度 & 產(chǎn)品資料
參考文獻(xiàn)

Cinacalcet metabolite M4 相關(guān)分類

  • 摩爾計(jì)算器

  • 稀釋計(jì)算器

The molarity calculator equation

Mass (g) = Concentration (mol/L) × Volume (L) × Molecular Weight (g/mol)

質(zhì)量   濃度   體積   分子量 *
= × ×

The dilution calculator equation

Concentration (start) × Volume (start) = Concentration (final) × Volume (final)

This equation is commonly abbreviated as: C1V1 = C2V2

濃度 (start) × 體積 (start) = 濃度 (final) × 體積 (final)
× = ×
C1   V1   C2   V2
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  • Do most proteins show cross-species activity?

    Species cross-reactivity must be investigated individually for each product. Many human cytokines will produce a nice response in mouse cell lines, and many mouse proteins will show activity on human cells. Other proteins may have a lower specific activity when used in the opposite species.

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產(chǎn)品名稱:
Cinacalcet metabolite M4
目錄號(hào):
HY-135601
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