TGX 221

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 1417

CAS [663619-89-4]

MF C21H24N4O2
MW 364.44

Purity: 99%
Soluble in DMSO

TGX 221

Description

Potent and specific PI3K p110β inhibitor

SP Jackson et al. PI 3-kinase p110b: A new target for antithrombotic therapy. Nature Medicine 2005, 11(5), 507-514.

BT Hennessy et al. Exploiting the PI3K/AKT pathway for cancer drug discovery. Nature Reviews Drug Discovery 2005, 4988-1004.

AM Condliffe et al. Sequential activation of class IB and class IA PI3K is important for the primed respiratory burst of human but not murine neutrophils. Blood 2005, 106, 1432-1440.

Cell Signaling & Oncology PI3K PI3K-Akt-mTOR EC 2.7.1.153

PI3K inhibitor (p110 β specific)

Chemical name

7-methyl-2-morpholin-4-yl-9-(1-phenylaminoethyl)-pyrido[1,2-a]-pyrimidin-4-one

Parent CAS No.

[663619-89-4]

Order

Size	Unit Price	Stock
2 mg	$77.00	In Stock
5 mg	$104.50	In Stock
25 mg	$368.50	In Stock

Special Offers

Size	Unit Price	Stock
2 x 5 mg	$154.00	In Stock
2 x 25 mg	$528.00	In Stock

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TGX 221

Description

Chemical name

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