UNC0638

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 1889

CAS [1255580-76-7]

MF C30H47N5O2
MW 509.73

Purity: 98%
Soluble in DMSO

UNC0638

Description

Potent and selective G9a (EHMT2)/GLP (EHMT1) inhibitor (G9a IC50: <15 nM; GLP IC50: 19 nM); chemical probe for G9a and GLP methyltransferase inhibition in cells

M Vedadi et al. A chemical probe selectively inhibits G9a and GLP methyltransferase activity in cells. Nat. Chem. Biol. 2011, 7(8), 566-574.

F Liu et al. Optimization of cellular activity of G9a inhibitors 7-aminoalkoxy-quinazolines. J. Med. Chem. 2011, 54(17), 6139-6150.

Apoptosis Cell Cycle Regulation Cell Signaling & Oncology Epigenetics EC 2.1.1.43 HMTase

Inhibitor of G9a (EHMT2)/GLP (EHMT1)

Chemical name

2-cyclohexyl-N-(1-isopropylpiperidin-4-yl)-6-methoxy-7-(3-(pyrrolidin-1-yl)propoxy)quinazolin-4-amine

Parent CAS No.

[1255580-76-7]

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Size	Unit Price	Stock
2 mg	$93.50	In Stock
5 mg	$137.50	In Stock
25 mg	$478.50	In Stock

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Size	Unit Price	Stock
2 x 5 mg	$198.00	In Stock
2 x 25 mg	$748.00	In Stock

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UNC0638

Description

Chemical name

Parent CAS No.

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