MK 5108 - VX 689

Based on 20 reference(s) in Google Scholar 80 100 20

Axon 1961

CAS [1010085-13-8]

MF C22H21ClFN3O3S
MW 461.94

Purity: 98%
Optical purity: Optically pure
Soluble in DMSO

MK 5108

Description

Highly potent and selective inhibitor of Aurora A kinase (AurA); MK5108 exhibits marked effects on the growth of tumor cells in vitro and in vivo; also enhances the antitumoractivity of Docetaxel without exacerbrating the toxicity in vivo

T Shimomura et al. MK-5108, a highly selective Aurora-A kinase inhibitor, shows antitumor activity alone and in combination with docetaxel. Mol. Cancer Ther. 2010, 9(1), 157-166.

Cell Cycle Regulation Cell Signaling & Oncology Epigenetics EC 2.7.11.1 Aurora

Inhibitor of Aurora A kinase

Chemical name

(1r,4r)-4-(3-chloro-2-fluorophenoxy)-1-((6-(thiazol-2-ylamino)pyridin-2-yl)methyl)cyclohexanecarboxylic acid

Parent CAS No.

[1010085-13-8]

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Size	Unit Price	Stock
5 mg	$121.00	In Stock
25 mg	$418.00	In Stock

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MK 5108 - VX 689

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成人免费xx,国产又黄又湿又刺激不卡网站,成人性视频app菠萝网站,色天天天天

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MK 5108 - VX 689

Description

Chemical name

Parent CAS No.

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