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Varenicline Tartrate
Catalog No.
A5391
Subtype-selective agonist of α4β2 nicotinic receptors,orally active
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Orally active, subtype-selective partial agonist at α4β2 nicotinic receptors (Ki values are 0.06, 240, 322 and 3540 nM for α4β2, α3β4, α7, α1βγδ receptors respectively). Reduces nicotine-evoked dopamine release in vitro and decreases nicotine self-adminis
| Physical Appearance | A solid |
| Storage | Store at -20°C |
| M.Wt | 361.35 |
| Cas No. | 375815-87-5 |
| Formula | C13H13N3·C4H6O6 |
| Solubility | insoluble in EtOH; ≥18.07 mg/mL in DMSO; ≥96.2 mg/mL in H2O |
| Chemical Name | (6R)-7,8,9,10-tetrahydro-6H-6,10-methanoazepino[4,5-g]quinoxaline (2R,3R)-2,3-dihydroxysuccinate |
| SDF | Download SDF |
| Canonical SMILES | O=C([C@]([C@@](C(O[H])=O)([H])O[H])([H])O[H])O[H].[H][C@@]12C([H])([H])C(C([H])([H])N([H])C2([H])[H])([H])C3=C([H])C4=NC([H])=C([H])N=C4C([H])=C13 |
| Shipping Condition | Small Molecules with Blue Ice, Modified Nucleotides with Dry Ice. |
| General tips | We do not recommend long-term storage for the solution, please use it up soon. |
Quality Control & MSDS
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Chemical structure
