Structure of Anidulafungin
CAS No.: 166663-25-8
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Anidulafungin is an echinocandin antifungal agent used to treat invasive Aspergillus infection, working by inhibiting (1→3)-β-D-glucan synthase, an enzyme important to the synthesis of the fungal cell wall.
Synonyms: LY303366; VER-002; VEchinocandin
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Batch number can be found on the product's label following the word 'Batch'.
Search for reports by entering the product batch number.
Batch number can be found on the product's label following the word 'Batch'.
Search for reports by entering the product batch number.
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CAS No. : | 166663-25-8 |
Formula : | C58H73N7O17 |
M.W : | 1140.24 |
SMILES Code : | OC1CC(C(NC(C(NC(C(N2C(C(NC(C(CC(C(NC(C3=O)C(C)O)=O)NC(C4=CC=C(C=C4)C5=CC=C(C=C5)C6=CC=C(C=C6)OCCCCC)=O)O)O)=O)C(C(C2)C)O)=O)C(O)C)=O)C(C(C7=CC=C(C=C7)O)O)O)=O)N3C1 |
Synonyms : |
LY303366; VER-002; VEchinocandin
|
MDL No. : | MFCD00917070 |
GHS Pictogram: |
![]() ![]() |
Signal Word: | Warning |
Hazard Statements: | H302-H319-H361 |
Precautionary Statements: | P264-P270-P301+P312-P330-P501-P305+P351+P338-P337+P313-P280-P201-P202-P281-P308+P313 |
In Vitro:
Cell Line
|
Concentration | Treated Time | Description | References |
African green monkey kidney cells (Vero) | 5, 10, 20 μM | 1 hour | Evaluate the inhibitory effect of Anidulafungin on SFTSV infection, results showed that Anidulafungin effectively inhibits SFTSV entry into cells. | PMC9585728 |
Candida glabrata | 0.01 to 0.1 mg/L | 24 h and 48 h | To determine the minimum inhibitory concentration (MIC) of Anidulafungin against Candida glabrata. Results showed that MIC values were identical at 24 and 48 hours, and for both 50% and ≥95% reduction in turbidity. | PMC1635198 |
Candida auris | 0.016 to 8 mg/L | 24 hours | Evaluate the in vitro synergistic activity of Anidulafungin in combination with manogepix or 5-flucytosine against Candida auris, showing synergistic effects | PMC10269148 |
Candida auris (South American clade) | 0.25, 1, 8, 16, 32 mg/L | 24 hours | Anidulafungin showed a negligible fungistatic effect against the isolates from Israel but was fungistatic against the environmental isolates. | PMC10222763 |
Candida auris (South African clade) | 0.25, 1, 8, 16, 32 mg/L | 24 hours | Anidulafungin produced a weak fungistatic effect against the South African clade isolates. | PMC10222763 |
Candida auris (East Asian clade) | 0.25, 1, 8, 16, 32 mg/L | 24 hours | Anidulafungin showed concentration-dependent killing activity against the type strain and fungistatic activity against the other isolates. | PMC10222763 |
Candida auris (South Asian clade) | 0.25, 1, 8, 16, 32 mg/L | 24 hours | Anidulafungin exhibited weak fungistatic activity against wild-type isolates and the isolate with a mutation in the hot-spot 2 region of FKS1 but was ineffective against the isolates with a mutation in the hot-spot 1 region. | PMC10222763 |
BV2 microglia cells | 1 μM | 24 hours | To evaluate the protective effect of Anidulafungin against Aβ oligomer-induced cytotoxicity. Results showed 1 μM Anidulafungin significantly attenuated AβO-induced cytotoxicity, restoring cell viability to 93.30% (vs. 68.66% with AβO alone). | PMC11342299 |
Candida auris clinical isolates | 0.06-4 μg/mL | 48 hours | Evaluate the antifungal effect of Anidulafungin in combination with citral, showing synergistic effects against 36.84% of isolates and additive effects against 57.89% | PMC10300739 |
In Vivo:
Species
|
Animal Model
|
Administration | Dosage | Frequency | Description | References |
Caenorhabditis elegans | C. elegans infection model | Liquid media | 0.06 and 0.25 μg/mL | Observed every 24 hours for 120 hours | Evaluate the in vivo antifungal effect of Anidulafungin in combination with citral, showing significantly increased survival rates of nematodes | PMC10300739 |
CD1 mice | Invasive aspergillosis model | Intraperitoneal injection | 1 and 5 mg/kg/day | Initiated 2 h post-infection, continued for 5 days (day 0 to day 4) | Assessed therapeutic efficacy of Anidulafungin alone and combined with amphotericin B. AFG (1 and 5 mg/kg/day) and combinations significantly prolonged survival, but combinations were not superior to monotherapy; 5 mg/kg/day reduced kidney fungal burden but was ineffective in brain tissues. | PMC2737837 |
Female outbred Swiss Webster mice | Neutropenic model of disseminated candidiasis | Intraperitoneal injection | 1 to 20 mg/kg | Single dose, observed at 24 h and 96 h | To evaluate the pharmacodynamics and pharmacokinetics of Anidulafungin in neutropenic mice. Results showed delayed peak concentrations in kidneys compared to serum, with a serum terminal half-life of 21.6 h. A single dose of ≥8 mg/kg resulted in a persistent decrease in kidney fungal burden over 96 h. | PMC1635198 |
A129 mice | SFTSV infection model | Intraperitoneal injection | 10 mg/kg | Once daily for 14 days | Evaluate the therapeutic effect of Anidulafungin on SFTSV-infected mice, results showed that Anidulafungin alleviates symptoms, reduces tissue lesions, and improves survival rates. | PMC9585728 |
Hairless mice | Candida albicans CNS infection model | Intraperitoneal injection | 10 mg/kg/day | Once daily for 8 days | To evaluate the efficacy of anidulafungin in treating Candida albicans CNS infection. Results showed that 10 mg/kg/day anidulafungin significantly reduced mortality and fungal burden in brain tissue, comparable to amphotericin B and superior to voriconazole. | PMC2715626 |
BALB/c male mice | Neutropenic mouse bloodstream infection model | Intraperitoneal | 5 mg/kg | Once daily for 6 days | To evaluate the in vivo efficacy of Anidulafungin against four Candida auris clades. Results showed that regardless of the isolate and clade, all echinocandin regimens significantly improved survival after 21 days (p=0.0041 to p<0.0001). Anidulafungin produced 1-4 log mean CFU/g decreases in the fungal kidney and heart burdens. | PMC11433204 |
Clinical Trial:
NCT Number | Conditions | Phases | Recruitment | Completion Date | Locations |
NCT01307930 | Obesity|Mycoses | PHASE4 | COMPLETED | 2025-11-12 | University of Texas Southweste... More >>rn Medical Center, Dallas, Texas, 75390, United States Less << |
NCT00537329 | Candidemia | PHASE3 | COMPLETED | 2025-03-09 | Pfizer Investigational Site, A... More >>hmedabad, Gujarat, 380 054, India|Pfizer Investigational Site, Bangalore, Karnataka, 560034, India|Pfizer Investigational Site, Mumbai, Maharashtra, 400 022, India|Pfizer Investigational Site, Ludhiana, Punjab, 141 001, India|Pfizer Investigational Site, Noida, Uttar Pradesh, 201301, India|Pfizer Investigational Site, Legaspi Village, Makati City, 1200, Philippines|Pfizer Investigational Site, Pan-Chiao, Taipei, 220, Taiwan|Pfizer Investigational Site, Taichung, 404, Taiwan|Pfizer Investigational Site, Tainan, 704, Taiwan|Pfizer Investigational Site, Taipei, 100, Taiwan|Pfizer Investigational Site, Pathumwan, Bangkok, 10330, Thailand|Pfizer Investigational Site, Amphoe Mueang, Chiang Mai, 50200, Thailand|Pfizer Investigational Site, Amphoe Mueang, Khon Kaen, 40002, Thailand Less << |
NCT01734525 | Candidemia | PHASE4 | COMPLETED | 2025-12-13 | Federal University of Rio de J... More >>aneiro, Rio de Janeiro, RJ, 21941913, Brazil Less << |
NCT00734500 | Invasive Fungal Infections | PHASE1 | COMPLETED | 2025-06-10 | Duke University, Durham, North... More >> Carolina, 27705, United States Less << |
NCT00058682 | Candida|Candidiasis | PHASE3 | COMPLETED | 2025-01-05 | National Cancer Institute (NCI... More >>), Bethesda, Maryland, 20892, United States Less << |
NCT00892359 | Acute Renal Failure|Infection | PHASE2 | UNKNOWN | - | Medical University of Vienna, ... More >>Vienna, 1090, Austria Less << |
NCT00056381 | Neutropenia | PHASE1|PHASE2 | COMPLETED | 2025-06-04 | Versicor, King of Prussia, Pen... More >>nsylvania, 19406, United States Less << |
NCT01053884 | Hematologic Malignancies | PHASE2 | TERMINATED | 2025-09-11 | Elisabethinen hospital, Linz, ... More >>Upper Austria, 4020, Austria Less << |
Bio Calculators | ||||
Preparing Stock Solutions | ![]() |
1mg | 5mg | 10mg |
1 mM 5 mM 10 mM |
0.88mL 0.18mL 0.09mL |
4.39mL 0.88mL 0.44mL |
8.77mL 1.75mL 0.88mL |
Tags: Anidulafungin | LY303366 | LY 303366 | LY-303366 | Fungal | Antibiotic | semisynthetic echinocandin | antifungal agent | 166663-25-8
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Code | Phrase |
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P232 | Protect from moisture. |
P233 | Keep container tightly closed. |
P234 | Keep only in original container. |
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P240 | Ground/bond container and receiving equipment. |
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P265 | Wash skin thouroughly after handling. |
P270 | Do not eat, drink or smoke when using this product. |
P271 | Use only outdoors or in a well-ventilated area. |
P272 | Contaminated work clothing should not be allowed out of the workplace. |
P273 | Avoid release to the environment. |
P280 | Wear protective gloves/protective clothing/eye protection/face protection. |
P281 | Use personal protective equipment as required. |
P282 | Wear cold insulating gloves/face shield/eye protection. |
P283 | Wear fire/flame resistant/retardant clothing. |
P284 | Wear respiratory protection. |
P285 | In case of inadequate ventilation wear respiratory protection. |
P231 + P232 | Handle under inert gas. Protect from moisture. |
P235 + P410 | Keep cool. Protect from sunlight. |
Response | |
Code | Phrase |
P301 | IF SWALLOWED: |
P304 | IF INHALED: |
P305 | IF IN EYES: |
P306 | IF ON CLOTHING: |
P307 | IF exposed: |
P308 | IF exposed or concerned: |
P309 | IF exposed or if you feel unwell: |
P310 | Immediately call a POISON CENTER or doctor/physician. |
P311 | Call a POISON CENTER or doctor/physician. |
P312 | Call a POISON CENTER or doctor/physician if you feel unwell. |
P313 | Get medical advice/attention. |
P314 | Get medical advice/attention if you feel unwell. |
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P321 | |
P322 | |
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P338 | Remove contact lenses, if present and easy to do. Continue rinsing. |
P340 | Remove victim to fresh air and keep at rest in a position comfortable for breathing. |
P341 | If breathing is difficult, remove victim to fresh air and keep at rest in a position comfortable for breathing. |
P342 | If experiencing respiratory symptoms: |
P350 | Gently wash with plenty of soap and water. |
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P362 | Take off contaminated clothing and wash before reuse. |
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P371 | In case of major fire and large quantities: |
P372 | Explosion risk in case of fire. |
P373 | DO NOT fight fire when fire reaches explosives. |
P374 | Fight fire with normal precautions from a reasonable distance. |
P376 | Stop leak if safe to do so. Oxidising gases (section 2.4) 1 |
P377 | Leaking gas fire: Do not extinguish, unless leak can be stopped safely. |
P378 | |
P380 | Evacuate area. |
P381 | Eliminate all ignition sources if safe to do so. |
P390 | Absorb spillage to prevent material damage. |
P391 | Collect spillage. Hazardous to the aquatic environment |
P301 + P310 | IF SWALLOWED: Immediately call a POISON CENTER or doctor/physician. |
P301 + P312 | IF SWALLOWED: call a POISON CENTER or doctor/physician IF you feel unwell. |
P301 + P330 + P331 | IF SWALLOWED: Rinse mouth. Do NOT induce vomiting. |
P302 + P334 | IF ON SKIN: Immerse in cool water/wrap in wet bandages. |
P302 + P350 | IF ON SKIN: Gently wash with plenty of soap and water. |
P303 + P361 + P353 | IF ON SKIN (or hair): Remove/Take off Immediately all contaminated clothing. Rinse SKIN with water/shower. |
P304 + P312 | IF INHALED: Call a POISON CENTER or doctor/physician if you feel unwell. |
P304 + P340 | IF INHALED: Remove victim to fresh air and Keep at rest in a position comfortable for breathing. |
P304 + P341 | IF INHALED: If breathing is difficult, remove victim to fresh air and keep at rest in a position comfortable for breathing. |
P305 + P351 + P338 | IF IN EYES: Rinse cautiously with water for several minutes. Remove contact lenses, if present and easy to do. Continue rinsing. |
P306 + P360 | IF ON CLOTHING: Rinse Immediately contaminated CLOTHING and SKIN with plenty of water before removing clothes. |
P307 + P311 | IF exposed: call a POISON CENTER or doctor/physician. |
P308 + P313 | IF exposed or concerned: Get medical advice/attention. |
P309 + P311 | IF exposed or if you feel unwell: call a POISON CENTER or doctor/physician. |
P332 + P313 | IF SKIN irritation occurs: Get medical advice/attention. |
P333 + P313 | IF SKIN irritation or rash occurs: Get medical advice/attention. |
P335 + P334 | Brush off loose particles from skin. Immerse in cool water/wrap in wet bandages. |
P337 + P313 | IF eye irritation persists: Get medical advice/attention. |
P342 + P311 | IF experiencing respiratory symptoms: call a POISON CENTER or doctor/physician. |
P370 + P376 | In case of fire: Stop leak if safe to Do so. |
P370 + P378 | In case of fire: |
P370 + P380 | In case of fire: Evacuate area. |
P370 + P380 + P375 | In case of fire: Evacuate area. Fight fire remotely due to the risk of explosion. |
P371 + P380 + P375 | In case of major fire and large quantities: Evacuate area. Fight fire remotely due to the risk of explosion. |
Storage | |
Code | Phrase |
P401 | |
P402 | Store in a dry place. |
P403 | Store in a well-ventilated place. |
P404 | Store in a closed container. |
P405 | Store locked up. |
P406 | Store in corrosive resistant/ container with a resistant inner liner. |
P407 | Maintain air gap between stacks/pallets. |
P410 | Protect from sunlight. |
P411 | |
P412 | Do not expose to temperatures exceeding 50 oC/ 122 oF. |
P413 | |
P420 | Store away from other materials. |
P422 | |
P402 + P404 | Store in a dry place. Store in a closed container. |
P403 + P233 | Store in a well-ventilated place. Keep container tightly closed. |
P403 + P235 | Store in a well-ventilated place. Keep cool. |
P410 + P403 | Protect from sunlight. Store in a well-ventilated place. |
P410 + P412 | Protect from sunlight. Do not expose to temperatures exceeding 50 oC/122oF. |
P411 + P235 | Keep cool. |
Disposal | |
Code | Phrase |
P501 | Dispose of contents/container to ... |
P502 | Refer to manufacturer/supplier for information on recovery/recycling |
Physical hazards | |
Code | Phrase |
H200 | Unstable explosive |
H201 | Explosive; mass explosion hazard |
H202 | Explosive; severe projection hazard |
H203 | Explosive; fire, blast or projection hazard |
H204 | Fire or projection hazard |
H205 | May mass explode in fire |
H220 | Extremely flammable gas |
H221 | Flammable gas |
H222 | Extremely flammable aerosol |
H223 | Flammable aerosol |
H224 | Extremely flammable liquid and vapour |
H225 | Highly flammable liquid and vapour |
H226 | Flammable liquid and vapour |
H227 | Combustible liquid |
H228 | Flammable solid |
H229 | Pressurized container: may burst if heated |
H230 | May react explosively even in the absence of air |
H231 | May react explosively even in the absence of air at elevated pressure and/or temperature |
H240 | Heating may cause an explosion |
H241 | Heating may cause a fire or explosion |
H242 | Heating may cause a fire |
H250 | Catches fire spontaneously if exposed to air |
H251 | Self-heating; may catch fire |
H252 | Self-heating in large quantities; may catch fire |
H260 | In contact with water releases flammable gases which may ignite spontaneously |
H261 | In contact with water releases flammable gas |
H270 | May cause or intensify fire; oxidizer |
H271 | May cause fire or explosion; strong oxidizer |
H272 | May intensify fire; oxidizer |
H280 | Contains gas under pressure; may explode if heated |
H281 | Contains refrigerated gas; may cause cryogenic burns or injury |
H290 | May be corrosive to metals |
Health hazards | |
Code | Phrase |
H300 | Fatal if swallowed |
H301 | Toxic if swallowed |
H302 | Harmful if swallowed |
H303 | May be harmful if swallowed |
H304 | May be fatal if swallowed and enters airways |
H305 | May be harmful if swallowed and enters airways |
H310 | Fatal in contact with skin |
H311 | Toxic in contact with skin |
H312 | Harmful in contact with skin |
H313 | May be harmful in contact with skin |
H314 | Causes severe skin burns and eye damage |
H315 | Causes skin irritation |
H316 | Causes mild skin irritation |
H317 | May cause an allergic skin reaction |
H318 | Causes serious eye damage |
H319 | Causes serious eye irritation |
H320 | Causes eye irritation |
H330 | Fatal if inhaled |
H331 | Toxic if inhaled |
H332 | Harmful if inhaled |
H333 | May be harmful if inhaled |
H334 | May cause allergy or asthma symptoms or breathing difficulties if inhaled |
H335 | May cause respiratory irritation |
H336 | May cause drowsiness or dizziness |
H340 | May cause genetic defects |
H341 | Suspected of causing genetic defects |
H350 | May cause cancer |
H351 | Suspected of causing cancer |
H360 | May damage fertility or the unborn child |
H361 | Suspected of damaging fertility or the unborn child |
H361d | Suspected of damaging the unborn child |
H362 | May cause harm to breast-fed children |
H370 | Causes damage to organs |
H371 | May cause damage to organs |
H372 | Causes damage to organs through prolonged or repeated exposure |
H373 | May cause damage to organs through prolonged or repeated exposure |
Environmental hazards | |
Code | Phrase |
H400 | Very toxic to aquatic life |
H401 | Toxic to aquatic life |
H402 | Harmful to aquatic life |
H410 | Very toxic to aquatic life with long-lasting effects |
H411 | Toxic to aquatic life with long-lasting effects |
H412 | Harmful to aquatic life with long-lasting effects |
H413 | May cause long-lasting harmful effects to aquatic life |
H420 | Harms public health and the environment by destroying ozone in the upper atmosphere |
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