GCN2-IN-7 NEW
| Price | $313 | $787 | $1320 |
| Package | 1mg | 5mg | 10mg |
| Min. Order: | |
| Supply Ability: | 10g |
| Update Time: | 2025-04-30 |
Product Details
| Product Name: GCN2-IN-7 | CAS No.: 2396465-33-9 |
| Purity: 99.12% | Supply Ability: 10g |
| Release date: 2025/04/30 |
Product Introduction
Bioactivity
| Name | GCN2-IN-7 |
| Description | GCN2-IN-7 is an orally active, potent and selective inhibitor of the environmental sensing protein GCN2 with anti-tumor activity and can be used to study melanoma. |
| In vitro | 600 nM GCN2-IN-7 alleviates myeloid-derived suppressive cells (MDSC)-related T cell suppression and restores T cell proliferation. [1] |
| In vivo | Twice daily oral gavage of 15 mg/kg GCN2-IN-7 for 17 days showed potent target binding activity at reasonable doses. Twice daily oral gavage of 50 mg/kg GCN2-IN-7 for 17 days inhibited tumor growth in an LL2 homozygous mouse tumor model. [1] |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
| Solubility Information | DMSO : 40 mg/mL(75.84 mM), Sonication is recommended. |
| Keywords | GCN2 |
| Inhibitors Related | MSU-42011 | BTdCPU | GP 1a | GSK2606414 | DNL343 | ISRIB (trans-isomer) | Azoramide | SHP099 | PERK-IN-4 | ATPγS tetralithium salt | CCT020312 | 4EGI-1 |
| Related Compound Libraries | Bioactive Compound Library | Bioactive Compounds Library Max |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
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United States- Since: 2011-01-07
- Address: 36 Washington Street, Wellesley Hill, MA
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