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CT52923 NEW

Price	$30	$43	$67
Package	2mg	5mg	10mg

Min. Order:
Supply Ability:	10g
Update Time:	2024-11-19

Product Details

Product Name: CT52923	CAS No.: 205256-55-9
Purity: 99.88%	Supply Ability: 10g
Release date: 2024/11/19

Product Introduction

Bioactivity

Name	CT52923
Description	CT52923 is a selective, orally active antagonist of platelet-derived growth factor receptor (PDGFR), functioning as an ATP-competitive inhibitor. It has versatile applications for researching pathological diseases such as atherosclerosis, glomerulonephritis, liver cirrhosis, pulmonary fibrosis, and cancer.
In vitro	CT52923 inhibits PDGFRs and stem cell factor receptors with IC50 values of 100 to 200 nM. CT52923（0.01-30 μ M； 24 h) blocks smooth muscle cell migration or fibroblast proliferation induced by platelet-derived growth factor, IC50 is 64 and 280 nM respectively [1].
In vivo	CT52923 (oral; 5,15,30 and 50 mg/kg; twice daily) significantly inhibits the formation of neointima after carotid artery injury in rats [1].
Storage	Shipping with blue ice.
Solubility Information	DMSO : 60 mg/mL (128.33 mM)
Keywords	CT 52923 \| CT-52923 \| CT52923
Inhibitors Related	Nintedanib \| Regorafenib monohydrate \| Imatinib Mesylate \| Sunitinib Malate \| Sorafenib \| Regorafenib \| Nintedanib esylate \| Sorafenib tosylate \| Lenvatinib mesylate \| Imatinib \| Pazopanib \| Axitinib
Related Compound Libraries	Anti-Lung Cancer Compound Library \| Bioactive Compound Library \| Membrane Protein-targeted Compound Library \| Tyrosine Kinase Inhibitor Library \| Kinase Inhibitor Library \| Inhibitor Library \| Bioactive Compounds Library Max \| Anti-Cancer Compound Library \| Anti-Cancer Active Compound Library

Company Profile Introduction

Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers. TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.