CB1R Allosteric modulator 3 NEW
Price | $35 | $81 | $139 |
Package | 1mg | 5mg | 10mg |
Min. Order: | |
Supply Ability: | 10g |
Update Time: | 2024-11-19 |
Product Details
Product Name: CB1R Allosteric modulator 3 | CAS No.: 2633686-36-7 |
Purity: 98.18% | Supply Ability: 10g |
Release date: 2024/11/19 |
Product Introduction
Bioactivity
Name | CB1R Allosteric modulator 3 |
Description | CB1R Allosteric modulator 3 is a potent CB1R modulator that inhibits cAMP and β-Arrestin and can be used for the study of obesity and nicotine addiction. |
In vitro | At a duration of 30 minutes and concentrations ranging from 0.10 nM to 10 μM, CB1R Allosteric modulator 3 (compound 44) exhibits potent inhibition of cAMP and β-Arrestin, with EC50 values of 0.018 μM and 1.241 μM, respectively [1].Due to the presence of small lipophilic functional groups on the ortho-position of the GAT211 site-III phenyl ring, CB1R Allosteric modulator 3 can enhance CB1R ago-PAM activity [1]. |
Storage | Shipping with blue ice. |
Solubility Information | DMSO : 80 mg/mL (212.29 mM), Sonication is recommended. |
Inhibitors Related | β-Caryophyllene | Bithionol | CB2 modulator 1 | Pregnenolone | Pregnenolone acetate | CB1 antagonist 2 | OMDM-5 | 2,3-Butanediol | Drinabant | AM281 |
Related Compound Libraries | Bioactive Compound Library | Membrane Protein-targeted Compound Library | Mitochondria-Targeted Compound Library | Bioactive Compounds Library Max | GPCR Compound Library |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
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- Since: 2011-01-07
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