Product Details
Product Name:
Balovaptan |
CAS No.:
1228088-30-9 |
Purity:
99.34% |
Supply Ability:
10g |
Release date:
2024/11/01 |
Product Introduction
Bioactivity
名稱 | Balovaptan |
描述 | Balovaptan (RG7314) is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for human (hV1a) and mouse (mV1a) receptors. It is used for the research of autism. |
體外活性 | Balovaptan (RG7314) is a highly potent and selective brain-penetrant vasopressin 1a (hV1a) receptor antagonist, with Kis of 1 and 39 nM for hV1a and mhV1a. It is used for the research of autism. Balovaptan shows >30000-fold selectivity for hV1a over hV2 receptors, 9891-fold selectivity over hOTR (human oxytocin receptor)[1]. |
存儲(chǔ)條件 | Powder: -20°C for 3 years | In solvent: -80°C for 1 year | Shipping with blue ice. |
溶解度 | DMSO : 62.5 mg/mL (152.47 mM), Sonication is recommended.
|
關(guān)鍵字 | RG 7314 | RG-7314 | Vasopressin Receptor | inhibit | Inhibitor | Balovaptan |
相關(guān)產(chǎn)品 | Atosiban acetate | Desmopressin acetate (16679-58-6 free base) | OPC-51803 | Felypressin acetate | d[Cha4]-AVP acetate(500170-27-4 free base) | Nelivaptan | TASP0390325 | d[Leu4,Lys8]-VP acetate | L-371,257 | Fuscoside | Conopressin S acetate(111317-90-9 free base) | Tolvaptan |
相關(guān)庫(kù) | 經(jīng)典已知活性庫(kù) | 兒童藥物庫(kù) | 膜蛋白靶向化合物庫(kù) | 抗癌臨床化合物庫(kù) | 藥物功能重定位化合物庫(kù) | 抑制劑庫(kù) | 臨床期小分子藥物庫(kù) | 已知活性化合物庫(kù) | GPCR靶點(diǎn)分子庫(kù) | 抗癌藥物庫(kù) |
Company Profile Introduction
Target Molecule Corp. (TargetMol) is a global high-tech enterprise, headquartered in Boston, MA, specializing in chemical and biological research product and service to meet the research needs of global customers.
TargetMol has evolved into one of the biggest global compound library and small molecule suppliers and a customer based on 40+ countries. TargetMol offers over 80 types of compound libraries and a wide range of high-quality research chemicals including inhibitors, activator, natural compounds, peptides, inhibitory antibodies, and novel life-science kits, for laboratory and scientific use. Besides, virtual screening service is also available for customers who would like to conduct the computer-aided drug discovery.
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Recommended supplier
Product name |
Price |
|
Suppliers |
Update time |
|
$60.00/5mg |
VIP3Y
|
TargetMol Chemicals Inc.
|
2024-11-01 |