Enzastaurin (LY317615)
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- $8 - $2268
- Product name: Enzastaurin (LY317615)
- CAS: 170364-57-5
- MF: C32H29N5O2
- MW: 515.6
- EINECS:
- MDL Number:MFCD11040980
- Synonyms:1H-Pyrrole-2,5-dione, 3-(1-methyl-1H-indol-3-yl)-4-(1-(1-(2-pyridinylmethyl)-4-piperidinyl)-1H-indol-3-yl)-;Unii-uc96G28eqf;Enzastaurin,Enzstataurin,LY317615,170364-57-5,1H-Pyrrole-2,5-dione, 3-;3-(1-Methyl-1H-indol-3-yl)-4-(1-(1-(2-pyridinylmethyl)-4-piperidinyl)-1H-indol-3-yl)-1H-pyrrole-2,5-dione;Enzastaurin ( LY317615 );Enzastaurine;LY317615 (Enzastaurin);LY317615/Enzstataurin
51 prices
Selected condition：
Brand
- AK Scientific
- Alfa Aesar
- Ambeed
- American Custom Chemicals Corporation
- ApexBio Technology
- Arctom
- Axon Medchem
- Biorbyt Ltd
- Cayman Chemical
- Chemenu
- ChemScene
- Crysdot
- CSNpharm
- DC Chemicals
- Matrix Scientific
- Sigma-Aldrich
- Tocris
- TRC
Package
- 1mg
- 5mg
- 50
- 1unit
- 10
- 10mg
- 20mg
- 25mg
- 50mg
- 100mg
- 200mg
- 10mM(in 1mL DMSO)
- 250mg
- 500MG
- 1g
- ManufacturerAK Scientific
- Product numberW3715
- Product descriptionEnzastaurin
- Packaging25mg
- Price$108
- Updated2021-12-16
- Buy
- ManufacturerAK Scientific
- Product numberW3715
- Product descriptionEnzastaurin
- Packaging200mg
- Price$380
- Updated2021-12-16
- Buy
- ManufacturerAlfa Aesar
- Product numberJ67480
- Product descriptionEnzastaurin, 99%
- Packaging10mg
- Price$152
- Updated2023-06-20
- Buy
- ManufacturerAlfa Aesar
- Product numberJ67480
- Product descriptionEnzastaurin, 99%
- Packaging25mg
- Price$280
- Updated2023-06-20
- Buy
- ManufacturerAlfa Aesar
- Product numberJ67480
- Product descriptionEnzastaurin, 99%
- Packaging50mg
- Price$500
- Updated2023-06-20
- Buy
- ManufacturerAmbeed
- Product numberA473249
- Product descriptionEnzastaurin 98+%
- Packaging1mg
- Price$8
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA473249
- Product descriptionEnzastaurin 98+%
- Packaging5mg
- Price$18
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA473249
- Product descriptionEnzastaurin 98+%
- Packaging10mg
- Price$27
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA473249
- Product descriptionEnzastaurin 98+%
- Packaging50mg
- Price$71
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA473249
- Product descriptionEnzastaurin 98+%
- Packaging100mg
- Price$106
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA473249
- Product descriptionEnzastaurin 98+%
- Packaging250mg
- Price$180
- Updated2021-12-16
- Buy
- ManufacturerAmbeed
- Product numberA473249
- Product descriptionEnzastaurin 98+%
- Packaging1g
- Price$467
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0005201
- Product descriptionENZASTAURIN 95.00%
- Packaging10MG
- Price$245.7
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0005201
- Product descriptionENZASTAURIN 95.00%
- Packaging50MG
- Price$1443.75
- Updated2021-12-16
- Buy
- ManufacturerAmerican Custom Chemicals Corporation
- Product numberAPI0005201
- Product descriptionENZASTAURIN 95.00%
- Packaging500MG
- Price$1963.5
- Updated2021-12-16
- Buy
- ManufacturerApexBio Technology
- Product numberA1670
- Product descriptionEnzastaurin(LY317615)
- Packaging1unit
- Price$28
- Updated2021-12-16
- Buy
| Manufacturer | Product number | Product description | Packaging | Price | Updated | Buy |
|---|---|---|---|---|---|---|
| AK Scientific | W3715 | Enzastaurin | 25mg | $108 | 2021-12-16 | Buy |
| AK Scientific | W3715 | Enzastaurin | 200mg | $380 | 2021-12-16 | Buy |
| Alfa Aesar | J67480 | Enzastaurin, 99% | 10mg | $152 | 2023-06-20 | Buy |
| Alfa Aesar | J67480 | Enzastaurin, 99% | 25mg | $280 | 2023-06-20 | Buy |
| Alfa Aesar | J67480 | Enzastaurin, 99% | 50mg | $500 | 2023-06-20 | Buy |
| Ambeed | A473249 | Enzastaurin 98+% | 1mg | $8 | 2021-12-16 | Buy |
| Ambeed | A473249 | Enzastaurin 98+% | 5mg | $18 | 2021-12-16 | Buy |
| Ambeed | A473249 | Enzastaurin 98+% | 10mg | $27 | 2021-12-16 | Buy |
| Ambeed | A473249 | Enzastaurin 98+% | 50mg | $71 | 2021-12-16 | Buy |
| Ambeed | A473249 | Enzastaurin 98+% | 100mg | $106 | 2021-12-16 | Buy |
| Ambeed | A473249 | Enzastaurin 98+% | 250mg | $180 | 2021-12-16 | Buy |
| Ambeed | A473249 | Enzastaurin 98+% | 1g | $467 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0005201 | ENZASTAURIN 95.00% | 10MG | $245.7 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0005201 | ENZASTAURIN 95.00% | 50MG | $1443.75 | 2021-12-16 | Buy |
| American Custom Chemicals Corporation | API0005201 | ENZASTAURIN 95.00% | 500MG | $1963.5 | 2021-12-16 | Buy |
| ApexBio Technology | A1670 | Enzastaurin(LY317615) | 1unit | $28 | 2021-12-16 | Buy |
Properties
Melting point :249-261℃
Boiling point :767.2±60.0 °C(Predicted)
Density :1.34
RTECS :UX9626850
Flash point :417.8℃
storage temp. :-20°C
solubility :DMSO: soluble10mg/mL, clear (warmed)
form :powder
pka :7.88±0.60(Predicted)
color :, light orange to dark orange-red
Stability :Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
Boiling point :767.2±60.0 °C(Predicted)
Density :1.34
RTECS :UX9626850
Flash point :417.8℃
storage temp. :-20°C
solubility :DMSO: soluble10mg/mL, clear (warmed)
form :powder
pka :7.88±0.60(Predicted)
color :, light orange to dark orange-red
Stability :Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months.
Safety Information
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| Signal word: | Warning | |||||||||||||||||||||
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Description
Enzastaurin is a potent inhibitor of PKCβ (IC50 = 6 nM), with modest selectivity over PKCα, PKCγ, and PKCε (IC50 = 39, 83, and 110 nM, respectively). At 3 μM, enzastaurin also inhibits signaling through the Akt pathway. It suppresses angiogenesis, induces apoptosis, and reduces proliferation of cultured tumor cells. Because of these effects, enzastaurin has potential antineoplastic activity.More related product prices
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