Boronic acid, B-[3-[[4-(3-thienyl)-1H-1,2,3-triazol-1-yl]methyl]phenyl]-
- CAS No.
- 2232877-85-7
- Chemical Name:
- Boronic acid, B-[3-[[4-(3-thienyl)-1H-1,2,3-triazol-1-yl]methyl]phenyl]-
- Synonyms
- KPC-2-IN-1;Boronic acid, B-[3-[[4-(3-thienyl)-1H-1,2,3-triazol-1-yl]methyl]phenyl]-
- CBNumber:
- CB411944171
- Molecular Formula:
- C13H12BN3O2S
- Molecular Weight:
- 285.13
- MDL Number:
- MOL File:
- 2232877-85-7.mol
Boronic acid, B-[3-[[4-(3-thienyl)-1H-1,2,3-triazol-1-yl]methyl]phenyl]- Chemical Properties,Uses,Production
Uses
KPC-2-IN-1, boronic acid derivative, is a potent KPC-2 inhibitor with Ki of 0.032 μM. KPC-2-IN-1 enhances the activity of cefotaxime in KPC-2 expressing E. coli. KPC-2-IN-1 exhibits well tolerated in human HEK-293 cells, which can be used for the study of E. coli resistance to β-lactam antibiotics[1][2].
References
[1] Zhou J, et al. Triazole-substituted phenylboronic acids as tunable lead inhibitors of KPC-2 antibiotic resistance. Eur J Med Chem. 2022 Jun 28;240:114571. DOI:10.1016/j.ejmech.2022.114571
[2] Zhou J, et al. Boronic acid inhibitors of the class A β-lactamase KPC-2. Bioorg Med Chem. 2018 Jul 15;26(11):2921-2927. DOI:10.1016/j.bmc.2018.04.055
Boronic acid, B-[3-[[4-(3-thienyl)-1H-1,2,3-triazol-1-yl]methyl]phenyl]- Preparation Products And Raw materials
Raw materials
Preparation Products
Boronic acid, B-[3-[[4-(3-thienyl)-1H-1,2,3-triazol-1-yl]methyl]phenyl]- Suppliers
Supplier | Tel | Country | ProdList | Advantage | |
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Biorbyt Ltd. | -- | info@biorbyt.com | CHINA | 6482 | 58 |
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Biorbyt Ltd. | 58 |