MDK-8650
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- CAS號(hào):
- 736048-65-0
- 英文名:
- PKC-theta inhibitor
- 英文別名:
- MDK-8650;PKC-theta inhibitor;N4-((4-(Aminomethyl)cyclohexyl)methyl)-5-nitro-N2-(2-(trifluoromethoxy)benzyl)pyrimidine-2,4-diamine;2,4-Pyrimidinediamine, N4-[[4-(aminomethyl)cyclohexyl]methyl]-5-nitro-N2-[[2-(trifluoromethoxy)phenyl]methyl]-
- 中文名:
- MDK-8650
- 中文別名:
- 化合物PKC-THETA INHIBITOR;PKC-THETA INHIBITOR (混旋的);N4-((4-(氨基甲基)環(huán)己基)甲基)-5-硝基-N2-(2-(三氟甲氧基)芐基)嘧啶-2,4-二胺
- CBNumber:
- CB64809360
- 分子式:
- C20H25F3N6O3
- 分子量:
- 454.45
- MOL File:
- 736048-65-0.mol
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MDK-8650化學(xué)性質(zhì)
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沸點(diǎn):
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597.1±60.0 °C(Predicted)
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密度:
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1.356±0.06 g/cm3(Predicted)
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儲(chǔ)存條件:
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Store at -20°C
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溶解度:
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DMSO : 62.5 mg/mL (137.53 mM)
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形態(tài):
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Solid
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酸度系數(shù)(pKa):
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10.27±0.29(Predicted)
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顏色:
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White to off-white
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MDK-8650性質(zhì)、用途與生產(chǎn)工藝
PKC-theta inhibitor (compound 20) 可抑制PKC-θ，IC50值為18 nM。
| Target | Value |
PKCθ
()
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18 nM
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MDK-8650
上下游產(chǎn)品信息
上游原料
下游產(chǎn)品
| 更新日期 | 產(chǎn)品編號(hào) | 產(chǎn)品名稱 | CAS編號(hào) | 包裝 | 價(jià)格 |
|---|
| 2024/11/08 | S6577 | MDK-8650
PKC-theta inhibitor | 736048-65-0 | 2mg | 1367.96元 |
| 2024/11/08 | HY-112681 | PKC-theta inhibitor | | 1 mg | 720元 |
736048-65-0, MDK-8650 相關(guān)搜索:
- 抑制劑
- 藥靶配體
- 對(duì)照品
- C20H25F3N6O3
- N4-((4-(氨基甲基)環(huán)己基)甲基)-5-硝基-N2-(2-(三氟甲氧基)芐基)嘧啶-2,4-二胺
- 化合物PKC-THETA INHIBITOR
- PKC-THETA INHIBITOR (混旋的)
- 736048-65-0
- N4-((4-(Aminomethyl)cyclohexyl)methyl)-5-nitro-N2-(2-(trifluoromethoxy)benzyl)pyrimidine-2,4-diamine
- 2,4-Pyrimidinediamine, N4-[[4-(aminomethyl)cyclohexyl]methyl]-5-nitro-N2-[[2-(trifluoromethoxy)phenyl]methyl]-
- PKC-theta inhibitor
- MDK-8650