88150-59-8
中文名稱
UK51656
英文名稱
2-[[2-(Carbamoylmethylamino)ethoxy]methyl]-4-(2-chlorophenyl)-1,4-dihydro-6-methylpyridine-3,5-dicarboxylic acid 3-ethyl 5-methyl ester
CAS
88150-59-8
分子式
C22H28ClN3O6
分子量
465.93
MOL 文件
88150-59-8.mol
88150-59-8 結(jié)構(gòu)式
基本信息
中文別名
化合物 T13250 英文別名
UK-516562-[[2-(Carbamoylmethylamino)ethoxy]methyl]-4-(2-chlorophenyl)-1,4-dihydro-6-methylpyridine-3,5-dicarboxylic acid 3-ethyl 5-methyl ester
3,5-Pyridinedicarboxylic acid, 2-[[2-[(2-amino-2-oxoethyl)amino]ethoxy]methyl]-4-(2-chlorophenyl)-1,4-dihydro-6-methyl-, 3-ethyl 5-methyl ester
常見問題列表
生物活性
UK51656 是一種 calcium 拮抗劑，IC50 值為 4 nM。靶點(diǎn)
IC50: 4 nM (calcium)
體內(nèi)研究
UK51656 has an elimination half-life of 4.7 h, which is consistent with its duration of action in the anesthetized dog. The effect of UK51656 on coronary vascular resistance, has markedly long durations, being over 5 h.