122752-15-2
中文名稱
DELTORPHIN I
英文名稱
DELTORPHIN I
CAS
122752-15-2
分子式
C37H52N8O10
分子量
768.86
MOL 文件
122752-15-2.mol
更新日期
2025/02/14 15:09:49
122752-15-2 結(jié)構(gòu)式
基本信息
中文別名
化合物DELTORPHIN I(TFA)D-ALA2] DELTORPHIN I-新皮啡肽
英文別名
Delt-iDELTORPHIN 1
DELTORPHIN C
DELTORPHIN I
Deltorphin Ⅰ
ala(2)-deltorphin
Deltorphin I(TFA)
[D-ALA2]DELTORPHIN I
deltorphin I, Ala(2)-
M.W. 768.87 C37H52N8O10
物理化學(xué)性質(zhì)
沸點(diǎn)1242.4±65.0 °C(Predicted)
密度1.284±0.06 g/cm3(Predicted)
儲(chǔ)存條件-15°C
溶解度Soluble to 0.40 mg/ml in 50% acetonitrile / water
酸度系數(shù)(pKa)4.19±0.10(Predicted)
形態(tài)粉末
顏色White to off-white
DELTORPHIN I價(jià)格(試劑級(jí))
| 報(bào)價(jià)日期 | 產(chǎn)品編號(hào) | 產(chǎn)品名稱 | CAS號(hào) | 包裝 | 價(jià)格 |
| 2025/02/08 | HY-P1336 | DELTORPHIN I Deltorphin I | 122752-15-2 | 1 mg | 504元 |
| 2025/02/08 | HY-P1336 | DELTORPHIN I Deltorphin I | 122752-15-2 | 5 mg | 1260元 |
| 2025/02/08 | HY-P1336 | Deltorphin I | 122752-15-2 | 10 mg | 1890元 |
常見問(wèn)題列表
生物活性
Deltorphin I 是一種高親和力的選擇性 δ-阿片受體 (δ-opioid receptor) 激動(dòng)劑。靶點(diǎn)
δ-opioid receptor
體內(nèi)研究
Twice daily administration of Deltorphin I (20μg/mouse) for 4 days produces tolerance to Deltorphin I analgesia, as shown by the decrease in the analgesic response. The peak analgesic response to Deltorphin I (20 μg/mouse) at 10 min after injections is decreased from 8.36±0.28 s (the 1st day) to 4.53±0.14 s (the 4th day) markedly. Concurrent treatment of Melatonin (0.5, 1 and 2.5 mg/kg) and Deltorphin I (20 μg/mouse) twice daily for 4 days can attenuate the tolerance to Deltorphin I analgesia (P<0.05, <0.05 and <0.05), and this effect is dose dependent.