1222097-72-4
中文名稱
S38093 鹽
英文名稱
s38093
CAS
1222097-72-4
分子式
C17H25ClN2O2
分子量
324.85
MOL 文件
1222097-72-4.mol
更新日期
2024/12/15 19:35:15
1222097-72-4 結構式
基本信息
中文別名
S38093 鹽S 38093 鹽酸鹽
化合物S 38093 HCL
英文別名
s38093S38093 HCl
S 38093 HydrochL
S 38093 Hydrochloride
S 38093
S38093
S-38093
S38093 HCL
應用領域
用途一
S38093 is an inverse agonist at histamine H3 receptors. S 38093 displays a moderate affinity for rat, mouse and human H3 receptors (Ki=8.8, 1.44 and 1.2μM, respectively) with no affinity for other histaminergic receptors. In cellular models, the compound was able to antagonize mice H3 receptors (KB=0.65μM) and to suppress cAMP decrease induced by an H3 agonist via human H3 receptors (KB=0.11μM).