Identification | Back Directory | [Name]
Pravadoline | [CAS]
92623-83-1 | [Synonyms]
WIN-48098 Pravadoline Pravadolina Pravadolinum Pravadoline [inn] Pravadoline(WIN 48098) WIN-48098 (Pravadoline) Pravadolinum [inn-latin] Pravadolina [INN-Spanish] (2-methyl-1-(2-morpholinoethyl) 3-(4-Methoxybenzoyl)-2-methyl-1-(2-morpholinoethyl)-1H-indole (4-methoxyphenyl)(2-methyl-1-(2-morpholinoethyl)-1H-indol-3-yl)methanone (4-Methoxyphenyl)-[2-methyl-1-(2-morpholin-4-ylethyl)indol-3-yl]methanone (4-Methoxyphenyl)(2-methyl-1-(2-(4-morpholinyl)ethyl)-1H-indol-3-yl)methanone Methanone, (4-methoxyphenyl)(2-methyl-1-(2-(4-morpholinyl)ethyl)-1H-indol-3-yl)- | [Molecular Formula]
C23H26N2O3 | [MDL Number]
MFCD00864378 | [MOL File]
92623-83-1.mol | [Molecular Weight]
378.46 |
Chemical Properties | Back Directory | [Melting point ]
104-105 °C(Solv: ethyl acetate (141-78-6); hexane (110-54-3)) | [Boiling point ]
553.1±50.0 °C(Predicted) | [density ]
1.18±0.1 g/cm3(Predicted) | [solubility ]
DMF: 5 mg/ml; DMSO: 5 mg/ml; DMSO:PBS (pH 7.2) (1:10): 0.1 mg/ml; Ethanol: 0.15 mg/ml | [form ]
Off-white solid. | [pka]
7.07±0.10(Predicted) |
Hazard Information | Back Directory | [Uses]
An antiinflammatory and analgesic drug. | [Uses]
Cannabinoid receptor agonist | [Biological Activity]
Pravadoline is a novel analgesic agent whose mechanism of action includes inhibition of cyclooxygenase and cannabinoid receptor agonist activity. |
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