Identification | Back Directory | [Name]
c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate | [CAS]
1647120-04-4 | [Synonyms]
Velmupressin acetate V2 receptor (V2R) agonist c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2 acetate | [Molecular Formula]
C44H64ClN11O10S2 | [MDL Number]
MFCD32068008 | [MOL File]
1647120-04-4.mol | [Molecular Weight]
1006.63 |
Hazard Information | Back Directory | [Uses]
Velmupressin (c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-d-Arg-NEt2) acetate is a potent, selective and short-acting peptidic V2 receptor (V2R) agonist with EC50s of 0.07 and 0.02 nM for hV2R and rV2R, respectively[1]. | [References]
[1] Wi?niewski K, et al. Discovery of Potent, Selective, and Short-Acting Peptidic V2 Receptor Agonists. J Med Chem. 2019 May 23;62(10):4991-5005. DOI:10.1021/acs.jmedchem.9b00132 |
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