| Identification | Back Directory | [Name]
Mps1-IN-5 | [CAS]
1443763-60-7 | [Synonyms]
CS-2060
Mps1-IN-5
Empesertib
BAY 1161909
BAY-1161909;BAY1161909
BAY-1161909 Empesertib
（Empesertib）BAY1161909
Benzeneacetamide, 4-fluoro-N-[4-[2-[[2-methoxy-4-(methylsulfonyl)phenyl]amino][1,2,4]triazolo[1,5-a]pyridin-6-yl]phenyl]-α-methyl-, (αR)- | [Molecular Formula]
C29H26FN5O4S | [MOL File]
1443763-60-7.mol | [Molecular Weight]
559.62 |
| Chemical Properties | Back Directory | [density ]
1.36±0.1 g/cm3(Predicted) | [storage temp. ]
Store at -20°C | [solubility ]
DMSO:67.5(Max Conc. mg/mL);120.62(Max Conc. mM) | [form ]
Solid | [pka]
13.71±0.70(Predicted) | [color ]
White to off-white |
| Hazard Information | Back Directory | [Uses]
Empesertib (BAY 1161909) is a potent Mps1 inhibitor, with an IC50 of < 1 nM. | [IC 50]
Mps1: 1 nM (IC50) | [storage]
Store at -20°C | [References]
[1] SCHULZE, Volker, et al. PRODRUG DERIVATIVES OF SUBSTITUTED TRIAZOLOPYRIDINES. WO2014198647A2 |
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