| Identification | Back Directory | [Name]
-NETA | [CAS]
115066-04-1 | [Synonyms]
?-NETA
N2)pyridinato-&kappa
[2-(5-Methyl-1H-pyrazol-3-yl-&kappa
3-2-propenyl)palladium Tetrafluoroborate
2-(α-Naphthoyl)ethyltrimethylammonium iodide
3-(Trimethylaminio)-1-(2-naphtyl)-1-propanone
3-(Trimethylaminio)-1-(1-naphtyl)-1-propanone | [Molecular Formula]
C16H20INO | [MDL Number]
MFCD00209857 | [MOL File]
115066-04-1.mol | [Molecular Weight]
369.25 |
| Hazard Information | Back Directory | [Biological Activity]
Originally identified as a substrate (ChA or choline)-noncompetitiveslowly reversible choline acetyltransferase inhibitor (human ChAT/BuChE/AChE IC50 = 88 nM/33.3 μM/48.6 μM; does not affect mAChRsAChEChECrATganglionic or skeletal muscular nAChRs)α-NETA is a fluorescent molecule (Ex 255 & 297 nm; Em 427 nm) also known for its trace amine-associated receptor 5 (TAAR5 EC50 = 150 nM) agonist and chemokine-like receptor-1 antagonist (IC50 = 375 nM; 7 nM chemerin-induced CMKLR1 β-ARR2 recruitment) potencies both in cultures and in animal disease models in vivo (3-20 mg/kg via ip. or sc. in rats & mice). |
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| Company Name: |
G-CLONE
|
| Tel: |
400-910-1997 17560619001 |
| Website: |
http://www.g-clone.com/ |
| Company Name: |
MedChemExpress
|
| Tel: |
021-58955995 |
| Website: |
www.medchemexpress.com |
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