| Identification | Back Directory | [Name]
E 2078 | [CAS]
103613-84-9 | [Synonyms]
66A-078
Methyl-L-Tyr-Gly-Gly-L-Phe-L-Leu-L-Arg-N2-methyl-L-Arg-D-Leu-NHEt
N-Methyl-L-Tyr-Gly-Gly-L-Phe-L-Leu-L-Arg-Nα-methyl-L-Arg-D-Leu-NHEt
(2R)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-5-(diaminomethylideneamino)-2-[[(2S)-2-[[(2S)-2-[[2-[[2-[[(2S)-3-(4-hydroxyphenyl)-2-(methylamino)propanoyl]amino]acetyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-4-methylpentanoyl]amino]pentanoyl]-met | [Molecular Formula]
C50H81N15O9 | [MOL File]
103613-84-9.mol | [Molecular Weight]
1036.27 |
| Hazard Information | Back Directory | [Uses]
(N-Me-Tyr1,N-Me-Arg7,D-Leu-NHEt8)-Dynorphin A (1-8) (E-2078), a stable Dynorphin A (1–8) (HY-P2159) analog, is a kappa opioid receptor (KOR) agonist[1]. | [IC 50]
κ Opioid Receptor/KOR | [References]
[1] Butelman ER, et al. Effects of E-2078, a stable dynorphin A(1-8) analog, on sedation and serum prolactin levels in rhesus monkeys. Psychopharmacology (Berl). 1999 Nov;147(1):73-80. DOI:10.1007/s002130051144 |
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